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Estrace appartient à la classe de médicaments appelée thérapie de remplacement d’œstrogène (ERT).L’œstrogène est une hormone produite par les ovaires, ses récepteurs spécifiques étant localisés dans des organes différents (dans l’utérus, le vagin, l’urètre, les glandes mammaires, le foie, l’hypothalamus, l’hypophyse). Cette hormone stimule le développement et la croissance des organes sexuels féminins à partir de l’âge de la puberté: l’utérus, les trompes de Fallope, le vagin, le stroma et les conduits des glandes mammaires, la pigmentation des mamelons et des organes génitaux, la formation des caractères sexuels femelles secondaires, la formation des épiphyses des os longs. L’œstrogène est responsable du rejet rapide et régulier de l’endomètre et des saignements, en concentrations élevées, il provoque une hyperplasie de l’endomètre, inhibe la lactation, ainsi que la résorption osseuse. Estrace est utilisé pour traiter les symptômes de la ménopause, lesquels incluent les bouffées de chaleur et la siccité vaginale, les brûlures et les irritations. Il est également utilisé pour le traitement du cancer chez les femmes et les hommes et l’ostéoporose.
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